Microwave-Induced Synthesis of Enantiopure β- Lactams
نویسندگان
چکیده
منابع مشابه
Access to enantiopure 4-substituted 1,5-aminoalcohols from phenylglycinol-derived δ-lactams: synthesis of Haliclona alkaloids.
LiNH2BH3-promoted reductive opening of 8-substituted phenylglycinol-derived oxazolopiperidone lactams leads to enantiopure 4-substituted-5-aminopentanols, which are used as starting building blocks in the synthesis of the Haliclona alkaloids haliclorensin C, haliclorensin, and halitulin (formal). The starting lactams are easily accessible by a cyclocondensation reaction of (R)-phenylglycinol wi...
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ژورنال
عنوان ژورنال: Modern Chemistry & Applications
سال: 2017
ISSN: 2329-6798
DOI: 10.4172/2329-6798.1000228